Understanding Intrinsic Warhead Reactivity and Cysteine Druggability in Covalent Drug Discovery

oleh: Chiara Borsari, Alexandra Ioana Corfu, Paola Conti

Format: Article
Diterbitkan: Swiss Chemical Society 2023-05-01

Deskripsi

Subjek

Covalent inhibitors; Druggable cysteines; Intrinsic reactivity; Rational Design; Warhead