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Understanding Intrinsic Warhead Reactivity and Cysteine Druggability in Covalent Drug Discovery
oleh: Chiara Borsari, Alexandra Ioana Corfu, Paola Conti
Format: | Article |
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Diterbitkan: | Swiss Chemical Society 2023-05-01 |
Deskripsi
Subjek
Covalent inhibitors; Druggable cysteines; Intrinsic reactivity; Rational Design; Warhead