Hasil Pencarian - Rudolf Andrys
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The Influence of Locality on Phenolic Profile and Antioxidant Capacity of Bud Extracts oleh Zuzana Kovalikova, Jan Lnenicka, Rudolf Andrys
Diterbitkan 2021-07-01Dapatkan teks lengkap
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1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy oleh Barbara Kaproń, Robert Czarnomysy, Mariusz Wysokiński, Rudolf Andrys, Kamil Musilek, Andrea Angeli, Claudiu T. Supuran, Tomasz Plech
Diterbitkan 2020-01-01Dapatkan teks lengkap
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Allogeneic Bone Impregnated with Biodegradable Depot Delivery Systems for the Local Treatment of Joint Replacement Infections: An In Vitro Study oleh Libor Prokes, Eva Snejdrova, Tomas Soukup, Jana Malakova, Vladislav Frolov, Jan Loskot, Rudolf Andrys, Tomas Kucera
Diterbitkan 2022-10-01Dapatkan teks lengkap
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Charged pyridinium oximes with thiocarboxamide moiety are equally or less effective reactivators of organophosphate-inhibited cholinesterases compared to analogous carboxamides oleh Zuzana Kohoutova, David Malinak, Rudolf Andrys, Jana Svobodova, Miroslav Psotka, Monika Schmidt, Lukas Prchal, Kamil Musilek
Diterbitkan 2022-12-01Dapatkan teks lengkap
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A Complex In Vitro Degradation Study on Polydioxanone Biliary Stents during a Clinically Relevant Period with the Focus on Raman Spectroscopy Validation oleh Jan Loskot, Daniel Jezbera, Zuzana Olmrová Zmrhalová, Martina Nalezinková, Dino Alferi, Krisztina Lelkes, Petr Voda, Rudolf Andrýs, Alena Myslivcová Fučíková, Tomáš Hosszú, Aleš Bezrouk
Diterbitkan 2022-02-01Dapatkan teks lengkap
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BODIPY-labelled acetylcholinesterase reactivators can be encapsulated into ferritin nanovehicles for enhanced bioavailability in the CNS oleh Eliska Prchalova, Martina Sukupova, David Malinak, Rudolf Andrys, Ladislav Sivak, Vladimir Pekarik, Adam Skarka, Jana Svobodova, Lukas Prchal, Lukas Fresser, Zbynek Heger, Kamil Musilek
Diterbitkan 2023-11-01Dapatkan teks lengkap
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Privileged multi-target directed propargyl-tacrines combining cholinesterase and monoamine oxidase inhibition activities oleh Zofia Chrienova, Eugenie Nepovimova, Rudolf Andrys, Rafael Dolezal, Jana Janockova, Lubica Muckova, Lenka Fabova, Ondrej Soukup, Patrik Oleksak, Martin Valis, Jan Korabecny, José Marco-Contelles, Kamil Kuca
Diterbitkan 2022-12-01Dapatkan teks lengkap
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10
Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators oleh David Malinak, Rafael Dolezal, Vendula Hepnarova, Miroslava Hozova, Rudolf Andrys, Petr Bzonek, Veronika Racakova, Jan Korabecny, Lukas Gorecki, Eva Mezeiova, Miroslav Psotka, Daniel Jun, Kamil Kuca, Kamil Musilek
Diterbitkan 2020-01-01Dapatkan teks lengkap
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Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer’s disease therapy oleh Irene Pachón-Angona, Bernard Refouvelet, Rudolf Andrýs, Helène Martin, Vincent Luzet, Isabel Iriepa, Ignacio Moraleda, Daniel Diez-Iriepa, María-Jesús Oset-Gasque, José Marco-Contelles, Kamil Musilek, Lhassane Ismaili
Diterbitkan 2019-01-01Dapatkan teks lengkap
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12
Pyridinium-2-carbaldoximes with quinolinium carboxamide moiety are simultaneous reactivators of acetylcholinesterase and butyrylcholinesterase inhibited by nerve agent surrogates oleh Hyun Myung Lee, Rudolf Andrys, Jakub Jonczyk, Kyuneun Kim, Avinash G. Vishakantegowda, David Malinak, Adam Skarka, Monika Schmidt, Michaela Vaskova, Kamil Latka, Marek Bajda, Young-Sik Jung, Barbara Malawska, Kamil Musilek
Diterbitkan 2021-01-01Dapatkan teks lengkap
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Acetylcholinesterase Inhibition of Diversely Functionalized Quinolinones for Alzheimer’s Disease Therapy oleh Óscar M. Bautista-Aguilera, Lhassane Ismaili, Mourad Chioua, Rudolf Andrys, Monika Schmidt, Petr Bzonek, María Ángeles Martínez-Grau, Christopher D. Beadle, Tatiana Vetman, Francisco López-Muñoz, Isabel Iriepa, Bernard Refouvelet, Kamil Musilek, José Marco-Contelles
Diterbitkan 2020-05-01Dapatkan teks lengkap
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Discovery of small molecule mechanistic target of rapamycin inhibitors as anti-aging and anti-cancer therapeutics oleh Zofia Chrienova, David Rysanek, Patrik Oleksak, Dorota Stary, Dorota Stary, Marek Bajda, Milan Reinis, Romana Mikyskova, Ondrej Novotny, Rudolf Andrys, Adam Skarka, Pavla Vasicova, Josef Novak, Martin Valis, Martin Valis, Kamil Kuca, Zdenek Hodny, Eugenie Nepovimova
Diterbitkan 2022-12-01Dapatkan teks lengkap
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Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition oleh Patrik Oleksak, Miroslav Psotka, Marketa Vancurova, Olena Sapega, Jana Bieblova, Milan Reinis, David Rysanek, Romana Mikyskova, Katarina Chalupova, David Malinak, Jana Svobodova, Rudolf Andrys, Helena Rehulkova, Vojtech Skopek, Pham Ngoc Lam, Jiri Bartek, Zdenek Hodny, Kamil Musilek
Diterbitkan 2021-01-01Dapatkan teks lengkap
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Structure-Guided Design of <i>N</i>-Methylpropargylamino-Quinazoline Derivatives as Multipotent Agents for the Treatment of Alzheimer’s Disease oleh Barbora Svobodova, Lenka Pulkrabkova, Dawid Panek, Anna Misiachna, Marharyta Kolcheva, Rudolf Andrys, Jiri Handl, Jan Capek, Pavlina Nyvltova, Tomas Rousar, Lukas Prchal, Vendula Hepnarova, Martina Hrabinova, Lubica Muckova, Daniela Tosnerova, Galina Karabanovich, Vladimir Finger, Ondrej Soukup, Martin Horak, Jan Korabecny
Diterbitkan 2023-05-01Dapatkan teks lengkap
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Amaryllidaceae Alkaloids of Norbelladine-Type as Inspiration for Development of Highly Selective Butyrylcholinesterase Inhibitors: Synthesis, Biological Activity Evaluation, and Do... oleh Abdullah Al Mamun, Filip Pidaný, Daniela Hulcová, Jana Maříková, Tomáš Kučera, Monika Schmidt, Maria Carmen Catapano, Martina Hrabinová, Daniel Jun, Lubica Múčková, Jiří Kuneš, Jiří Janoušek, Rudolf Andrýs, Lucie Nováková, Rozálie Peřinová, Negar Maafi, Ondřej Soukup, Jan Korábečný, Lucie Cahlíková
Diterbitkan 2021-08-01Dapatkan teks lengkap
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Frentizole derivatives with mTOR inhibiting and senomorphic properties oleh Zofia Chrienova, David Rysanek, Josef Novak, Pavla Vasicova, Patrik Oleksak, Rudolf Andrys, Adam Skarka, Jelena Dumanovic, Zoran Milovanovic, Vesna Jacevic, Marketa Chvojkova, Kristina Holubova, Karel Vales, Veronika Skoupilova, Marian Valko, Klaudia Jomova, Suliman Y. Alomar, Fernanda D. Botelho, Tanos C.C. Franca, Kamil Kuca, Zdenek Hodny, Eugenie Nepovimova
Diterbitkan 2023-11-01Dapatkan teks lengkap
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