Hasil Pencarian - Giusy Tassone
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Structural Basis of Parasitic HSP90 ATPase Inhibition by Small Molecules oleh Giusy Tassone, Marco Mazzorana, Cecilia Pozzi
Diterbitkan 2022-10-01
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Metal Ion Binding to Human Glutaminyl Cyclase: A Structural Perspective oleh Giusy Tassone, Cecilia Pozzi, Stefano Mangani
Diterbitkan 2024-07-01
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Dynamic Interplay between Copper Toxicity and Mitochondrial Dysfunction in Alzheimer’s Disease oleh Giusy Tassone, Arian Kola, Daniela Valensin, Cecilia Pozzi
Diterbitkan 2021-04-01
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Structural Comparison of <i>Enterococcus faecalis</i> and Human Thymidylate Synthase Complexes with the Substrate dUMP and Its Analogue FdUMP Provides Hints about Enzyme Conformati... oleh Cecilia Pozzi, Stefania Ferrari, Rosaria Luciani, Giusy Tassone, Maria Paola Costi, Stefano Mangani
Diterbitkan 2019-03-01
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Structural Characterization of Human Heat Shock Protein 90 N-Terminal Domain and Its Variants K112R and K112A in Complex with a Potent 1,2,3-Triazole-Based Inhibitor oleh Giusy Tassone, Marco Mazzorana, Stefano Mangani, Elena Petricci, Elena Cini, Giuseppe Giannini, Cecilia Pozzi, Samuele Maramai
Diterbitkan 2022-08-01
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Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design oleh Tommaso Palomba, Giusy Tassone, Carmine Vacca, Matteo Bartalucci, Aurora Valeri, Cecilia Pozzi, Simon Cross, Lydia Siragusa, Jenny Desantis
Diterbitkan 2022-11-01
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Evidence of Pyrimethamine and Cycloguanil Analogues as Dual Inhibitors of <i>Trypanosoma brucei</i> Pteridine Reductase and Dihydrofolate Reductase oleh Giusy Tassone, Giacomo Landi, Pasquale Linciano, Valeria Francesconi, Michele Tonelli, Lorenzo Tagliazucchi, Maria Paola Costi, Stefano Mangani, Cecilia Pozzi
Diterbitkan 2021-06-01
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Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy oleh Giusy Tassone, Samuele Maramai, Marco Paolino, Stefania Lamponi, Federica Poggialini, Elena Dreassi, Elena Petricci, Stefano Alcaro, Cecilia Pozzi, Isabella Romeo
Diterbitkan 2024-09-01
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Chemically stable inhibitors of 14-3-3 protein–protein interactions derived from BV02 oleh Leire Iralde-Lorente, Ylenia Cau, Letizia Clementi, Lorenzo Franci, Giusy Tassone, Daniela Valensin, Mattia Mori, Adriano Angelucci, Mario Chiariello, Maurizio Botta
Diterbitkan 2019-01-01
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Small Molecules as Potential Inhibitors of the 14-3-3/c-Abl Interaction for the Treatment of CML oleh Leire Iralde-Lorente, Giusy Tassone, Ylenia Cau, Claire Munier, Lorenzo Franci, Cecilia Pozzi, Adriano Angelucci, Mario Chiariello, Matthew Perry, Stefano Mangani, Maurizio Botta
Diterbitkan 2019-08-01
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